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2017年重点实验室SCI/EI论文
2018-01-28   点击:[]

附表1:2017年重点实验室SCI/EI论文汇总表

序号

论文名称

SCIEI索引、收录

第一作者

通讯作者

期刊名称

1

Mitochondria-dependent benzothiadiazole-based molecule probe for quantitatively intracellular pH imaging.Dyes and Pigments

SCI    I

韩晓

郑一超

Dyes and Pigments

2

Synthesis and bioactivities study of new antibacterial peptide mimics: the dialkyl cationic amphiphiles

SCI    I

张恩

张恩,秦上尚,刘宏民

Eur. J. Med. Chem.

3

OP16, a novel ent-kaurene diterpenoid, potentiates the antitumor effect  of rapamycin by inhibiting rapamycin-induced feedback activation of Akt signaling in esophageal squamous cell carcinoma

SCI    I

彭柯峥

侯桂琴,

鲁照明

Biochemical Pharmacology

4

LPE-1, an orally active pyrimidine derivative, inhibits growth and mobility of human esophageal cancers by targeting LSD1

SCI    I

王博,赵兵,庞路平

余斌,马立英,刘宏民

Pharmacological Research

5

An Overview on Screening Methods for Lysine Specific Demethylase 1 (LSD1) Inhibitors

SCI    I

郑一超

余斌,

刘宏民

Current Medicinal Chemistry

6

Pro-apoptotic effects of JDA-202, a novel natural diterpenoid, on esophageal cancer through targeting peroxiredoxin I

SCI    I

石晓静,丁丽娜,周文娟

可钰,赵文,刘宏民

Antioxidants & Redox Signaling

7

Design, synthesis and antiproliferative activity of thiazolo[5,4-d]pyrimidine derivatives through the atom replacement strategy

SCI    I

李中华,

刘雪琪

余斌,

刘宏民

European Journal of Medicinal Chemistry

8

Identification of thiazolo[5,4-d]pyrimidine derivatives as potent antiproliferative agents through the drug repurposing strategy

SCI    I

李中华

余斌,

刘宏民

European Journal of Medicinal Chemistry

9

Synthesis, cytotoxic activity evaluation of novel1,2,3-triazole linked quinazoline derivatives

SCI    I

李中华

郑一超,

刘宏民

ACS Medicinal Chemistry Letters

10

Discovery of resveratrol derivatives as novel LSD1 inhibitors: Design, synthesis and their biological evaluation

SCI    I

段迎超

郑一超,

刘宏民

European Journal of Medicinal Chemistry

11

Structure-Activity Relationship Studies of β-Lactam-azide Analogues as Orally Antitumor Agents Binding to Tubulin Colchicine Site

SCI    I

付冬君,

符玲

张雁冰,

刘宏民

Scientific Reports

12

Discovery of 5,6-diaryl-1,2,4-triazines hybrids as potential apoptosis inducers

SCI    I

付冬君

张赛扬,张雁冰,刘宏民

European Journal of Medicinal Chemistry

13

Gene expression profiling and pathway network analysis of anti-tumor activity by Jaridon 6 in esophageal cancer

SCI    I

符玲

可钰,

刘宏民

European Journal of Pharmacology

14

Design, synthesis and biological evaluation of [1,2,4]triazolo[1,5-a]pyrimidines as potent lysine specific demethylase 1 (LSD1/KDM1A) inhibitors

SCI    I

王帅,

赵丽杰

余斌,

刘宏民

European Journal of Medicinal Chemistry

15

Advances toward LSD1 inhibitors for cancer therapy

SCI    I

付晓丽

余斌

Future Medicinal Chemistry

16

Design and synthesis of formononetin-dithiocarbamate hybrids that inhibit growth and migration of PC-3 cells via MAPK/Wnt signaling pathways.

SCI    I

付冬君

张雁冰

Eur. J. Med. Chem.

17

NOTA Analogue: a First Dithiocarbamate Inhibitor of Metallo-β-lactamases

SCI    II

张恩

张恩,肖春玲,秦上尚

Bioorg. Med. Chem. Lett.

18

Design, synthesis and preliminary antiproliferative activity studies of new diheteroaryl thioether derivatives

SCI    II

李中华

余斌,刘宏民

Bioorganic & Medicinal Chemistry Letters

19

3D-QSAR (CoMFA, CoMSIA), molecular docking and molecular dynamics simulations study of 6-aryl-5-cyano-pyrimidine derivatives as potential LSD1 inhibitors

SCI   II

丁丽娜

李雯,刘宏民

Bioorganic & Medicinal Chemistry Letters

20

Jesridonin in Combination with Paclitaxel Demonstrates Synergistic Anti-tumor Activity in Human Esophageal Carcinoma Cells

SCI    II

王淙

可钰,刘宏民

Bioorganic & Medicinal Chemistry Letters

21

Single-Step Multiresidue Determination of β-Lactam Antibiotics and β-Agonists in Porcine Muscle by Liquid Chromatography-Tandem Mass Spectrometry

SCI    II

李娟

刘宏民,张雁冰

Food Analytical Methods

22

Design, synthesis, and biological evaluation of new thiazolo[5,4-d]pyrimidine derivatives as potent antiproliferative agents

SCI   II

李中华,

刘雪琪

余斌,刘宏民

MedChemComm

23

diversity of phenothiazines: design and synthesis of phenothiazine-dithiocarbamate hybrids as potential cell-cycle blockers

SCI    II

付冬君

张赛扬,张雁冰,刘宏民

Molecular Diversity

24

Thiosemicarbazone-based selective proliferation inactivators inhibit gastric cancer cell growth, invasion, and migration

SCI    II

户彪,王博,赵兵

马立英,刘宏民

MedChemComm

25

Baicalin, a natural LSD1 inhibitor

SCI   II

郑一超

刘宏民

Bioorganic Chemistry

26

A General Asymmetric Synthesis of (R)-Matsutakeol and Flavored Analogs

SCI    II

刘佳

那日松,余斌

Molecules

27

Discovery of tranylcypromine analogs with an acylhydrazone
substituent as LSD1 inactivators: Design, synthesis and their biological
evaluation

SCI    II

孙凯

刘宏民,郑一超

Bioorganic & Medicinal Chemistry Letters

28

A novel chalcone derivative S17 induces apoptosis through ROS dependent DR5 up-regulation in gastric cancer cells.

SCI    II

张赛扬、李婷玉

徐洪德、金成允

Scientific Reports

29

One-pot synthesis of soluble and fluorescent aliphatic hyperbranched poly(amide-imide) with solventdependent emission,

SCI   II

王荣荣

李雯

Journal of Polymer Science Part A Polymer Chemistry,

30

Asymmetric Synthesis and Antitumor Activity of Spiro-Oxadiazole Derivatives from 1,4:3,6-Dianhydro-D-fructose

SCIE   Ⅴ区

丰五 

刘丰五

Chin. J. Chem.

31

Facile Approaches to 2-Deoxy-D-glucose and 2-Deoxy-α-D-glucopyranonucleosides from D-Glucal

SCI    III

刘丰五 

刘丰五

Synthesis

32

3-epi-Jaspine B类似物的合成和抗肿瘤活性评价

SCI    III

张恩

张恩,王亚娜

有机化学

33

Wild-type phosphatase and tensin homolog deleted on chromosome 10 improved the sensitivity of cells to rapamycin through regulating phosphorylation of Akt in esophageal squamous cell carcinoma

SCIE  Ⅴ区

鲁照明

侯桂琴

Dis Esophagus

34

Pharmacokinetics study of Zr-89-labeled melanin nanoparticle iniron-overload mice

SCIE   III

张朋俊

李晓天

Nuclear Medicine and Biology

35

核外氮杂甾体的合成及其抗肿瘤活性研究进展

SCI     III

余斌

刘宏民

有机化学

36

Synthesis and Antitumor Evaluation of 3-epi-Jaspine B Analogues

SCI    III

张恩

刘宏民

有机化学

37

Anti-proliferative effect of Jesridonin on paclitaxel-resistant EC109 human esophageal carcinoma cells

SCI   III

王淙

可钰,

刘宏民

International Journal of Biological Macromolecules

38

Geridonin, a novel derivative of oridonin, inhibits proliferation of MGC 803 cells both in vitro and in vivo through elevating the intracellular ROS

SCI   III

王赛琪,

王淙

可钰,

刘宏民

Journal of Pharmacy and Pharmacology

39

Sesquiterpenoids of Illicium jiadifengpi and Their Effects on
NGF-induced Neurite Outgrowth in PC12 Cells

SCIE

柳继锋

柳继锋

Chinese Journal of Chemistry

40

Design, synthesis and antiproliferative effect of 17β-amide derivatives of 2-methoxyestradiol and their studies on pharmacokinetics.

SCI    III

施秀芳

张振中

、王淙

Steroids

41

Effect of silybin on the fibrillation of hen egg-white lysozyme

SCIE

曾华金

杨冉

Journal of Molecular Recognition

42

Effect of nitrogen-doped graphene quantum dots on the fibrillation of hen egg-white lysozyme

SCIE

曾华金

杨冉

International Journal of Biological Macromolecules

43

Synthesis, Cytotoxic Activity Evaluation of Novel 1,2,3-Triazole
Linked Quinazoline Derivatives

SCIE

宋攀攀

张秋荣

Chin. J. Chem.

44

2,4,6-三取代嘧啶衍生物的合成及体外抗肿瘤活性研究

SCIE

宋攀攀

张秋荣

有机化学

45

1-苯基-4-取代酞嗪衍生物合成及抗肿瘤活性评价

SCIE

辛景超

张秋荣

有机化学

46

Immune-stimulating Effects of Mycoleptodonoides aitchisonii water extract via TNF-a and IFN-g

SCI   Ⅴ区

徐洪德

Dae-Hun Park

International Journal of Medicinal Mushrooms

47

Targeting the Bcl-2 family and P-glycoprotein reverses paclitaxel resistance in human esophageal carcinoma cell line.

SCIE

石晓丽

王淙

Biomed Pharmacother.

48

Bone morphogenetic protein 4 is overexpressed in and promotes migration and invasion of drug-resistant cancer cells.

SCIE

周凯瑞

王淙

Int J Biol Macromol.

49

Cepharanthine hydrochloride reverses P-glycoproteinmediated multidrug resistance in human ovarian carcinoma A2780/Taxol cells by inhibiting the PI3K/Akt signaling pathway

SCI    III

王亚峰

王庆端

Oncology Reports

50

Design, synthesis, antibacterial and insecticidal activities of novel N-phenylpyrazole fraxinellone hybrid compounds.

SCI    III

郭勇

郭勇

RSC Advances

51

Design, synthesis, and antibacterial activity of novel 8-methoxyquinoline-2-carboxamide compounds containing 1, 3, 4-thiadiazole moiety

SCI    III

曲来亮

郭勇

Zeitschrift für Naturforschung C



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药物关键制备技术教育部重点实验室

河南省郑州市高新区药物研究院203

0371-67781894,xhwei01@126.com